Dimenhydrinate
/api/v1/drug/dimenhydrinateMechanism of action
Sourced from openFDAMechanism-of-action class: Histamine H1 Receptor Antagonists.
Indications
Sourced from openFDA- Uses for prevention and treatment of these symptoms associated with motion sickness: nausea vomiting dizzinessICD-10: R11.2
Dosage & administration
Sourced from openFDADirections to prevent motion sickness, the first dose should be taken one-half to one hour before starting activity adults and children 12 years and over 1 to 2 tablets every 4-6 hours; do not exceed 8 tablets in 24 hours, or as directed by a doctor children 6 to under 12 years 1/2 to 1 tablet every 6-8 hours; do not exceed 3 tablets in 24 hours, or as directed by a doctor children 2 to under 6 years 1/2 tablet every 6-8 hours; do not exceed 1&1/2 tablets in 24 hours, or as directed by a doctor
Warnings & precautions
Sourced from openFDADo not use for children under 2 years of age unless directed by a doctor. Ask a doctor before use if you have a breathing problem such as emphysema or chronic bronchitis glaucoma difficulty in urination due to enlargement of the prostate gland Ask a doctor or pharmacist before use if you are taking sedatives or tranquilizers. When using this product marked drowsiness may occur alcohol, sedatives, and tranquilizers may increase drowsiness use caution when driving a motor vehicle or operating machinery avoid alcoholic beverages If pregnant or breast-feeding, ask a health professional before use. Keep out of reach of children. In case of overdose, get medical help or contact a Poison Control Center right away.
Approval history
Sourced from openFDA- Jun 23, 2004ANDAANDA040519Fresenius Kabi Usa
FAERS reports
- 1Nausea2,42123%
- 2Fatigue1,80617%
- 3Off Label Use1,75917%
- 4Headache1,54115%
- 5Vomiting1,35713%
- 6Malaise1,19411%
- 7Dizziness1,10811%
- 8Diarrhoea1,09811%
- 9Pain1,09110%
- 10Drug Ineffective1,08310%
- 11Pyrexia9669.3%
- 12Cough9168.8%
- 13Dyspnoea9138.8%
- 14Arthralgia8748.4%
- 15Rash8748.4%
Literature
Recent PubMed references pinned to Dimenhydrinate as a MeSH major topic. Citations link to pubmed.ncbi.nlm.nih.gov.
- Development and characterisation of fast dispersible dimenhydrinate tablets: Compactional study and in-silico PBPK modeling.PloS one · 2025 · Maqbool U, Zafar F, Yasmin R, et al.PMID 41144537DOI 10.1371/journal.pone.0334421
- Efficacy and safety of the cinnarizine/dimenhydrinate combination versus betahistine in the treatment of vertigo: A systematic literature review.Acta otorrinolaringologica espanola · 2025 · Martín-Enguix D, Gómez Gabaldón N, Amaro-Gahete FJ, et al.PMID 41038567DOI 10.1016/j.otoeng.2025.512274
- Design, Molecular Docking, In Vitro and In Vivo Evaluation of Dimenhydrinate-Cyclodextrin Complex for Fast Disintegrating Tablet.Current pharmaceutical design · 2026 · Samara RK, Sammour RMF, Seidel V, et al.PMID 40525446DOI 10.2174/0113816128398157250610113637
- Effects of Dimenhydrinate on Motor Behavior and Vascular Function: Possible Implications for the Field of Sports.Drug testing and analysis · 2025 · Flores-Monroy J, Ramírez-Hernández D, Lezama-Martínez D, et al.PMID 40049629DOI 10.1002/dta.3875
- ChlorTox scale assessment, greenness, and whiteness evaluation of selective spectrophotometric analysis of dimenhydrinate and cinnarizine.Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy · 2024 · Morgan EM, Fayez YM, Boltia SA, et al.PMID 38963943DOI 10.1016/j.saa.2024.124740
- Preparation, characterization, and in vitro cytogenotoxic evaluation of a novel dimenhydrinate-β-cyclodextrin inclusion complex.Biomolecules & biomedicine · 2024 · Hindija L, Hadžiabdić J, Haverić A, et al.PMID 38819319DOI 10.17305/bb.2024.10507
- Chronic high-dose dimenhydrinate use contributing to early multifactorial cognitive impairment.BMJ case reports · 2024 · Fabiano N, Dholakia S, Walker LAS, et al.PMID 38453220DOI 10.1136/bcr-2023-258493
- Acute Inhibition of the Human Kv1.5 Channel by H(1) Receptor Antagonist Dimenhydrinate: Mode of Action.Biological & pharmaceutical bulletin · 2023 · Park SI, Hwang S, Kim JH, et al.PMID 37779040DOI 10.1248/bpb.b23-00170
Clinical trials
The 10 most recently updated of 220 ClinicalTrials.gov registrations naming Dimenhydrinate as an intervention. Registration is not evidence of efficacy or safety — reference crosswalk only.
- Effectiveness and Safety of a Hydrating Gel Containing Polyvinyl Pyrrolidine, Algin and Hyaluronic Acid Applied After and Without Fractional CO₂ Laser TherapyNot yet recruiting · Interventional · 51 enrolled · Dr.dr.Irma Bernadette, SpKK (K)NCT07639151updated 2026-06-10
- Time Restricted Eating to Mitigate Obesity in Veterans With Spinal Cord InjuryEnrolling by invitation · Interventional · 15 enrolled · VA Office of Research and DevelopmentNCT05921487updated 2026-06-04
- Efficacy of Adjunctive Theravex Tissue Care® With Xenograft in Internal Sinus LiftingNot yet recruiting · Interventional · 16 enrolled · Ain Shams UniversityNCT07627633updated 2026-06-04
- Efficacy Test of a Moisturizing and Anti-aging Facial MaskActive not recruiting · Interventional · 60 enrolled · TCI Co., Ltd.NCT07622160updated 2026-06-03
- Observational Study of OROSEDAL in Sore Throat and Minor Oral LesionsRecruiting · Observational · 124 enrolled · Laboratoires ElerteNCT07620353updated 2026-06-02
- Recommendations of Enhanced Recovery Interventions for Patient's Clinical Team and Collection of Associated DataCompleted · Phase 3 · Interventional · 3,395 enrolled · Jennifer Holder-MurrayNCT04606264updated 2026-05-28
- Evaluation of the Effect of the Toothpaste on Delicate GumsRecruiting · Interventional · 60 enrolled · Lacer S.A.NCT07494747updated 2026-05-14
- Effect of Neurodynamic Mobilization of Vagus Nerve on Irritable Bowel Syndrome in WomenNot yet recruiting · Interventional · 32 enrolled · Cairo UniversityNCT07560345updated 2026-05-07
- Porcine Derma for Soft Tissue Augmentation Around ImplantsEnrolling by invitation · Interventional · 15 enrolled · Universidade do PortoNCT07436091updated 2026-05-05
- Improving the Care of Incontinence-Associated Dermatitis (IAD) Using a Beta-Glucan Cream as a Hydrating and Soothing AgentNot yet recruiting · Interventional · 60 enrolled · University of AlbertaNCT07524439updated 2026-04-28
Frequently asked questions
- How does Dimenhydrinate work?
- Mechanism-of-action class: Histamine H1 Receptor Antagonists.
- What is Dimenhydrinate used for?
- According to FDA labeling, Dimenhydrinate carries indications including: Uses for prevention and treatment of these symptoms associated with motion sickness: nausea vomiting dizziness. This is a reference summary of labeled uses, not medical advice or a treatment recommendation.
- What class of drug is Dimenhydrinate?
- Dimenhydrinate is classified as Aminoalkyl ethers, Histamine H1 Receptor Antagonists, Decreased Histamine Activity.
- What are the brand names for Dimenhydrinate?
- Dimenhydrinate is marketed under brand names including Airmit, Dramamine, Driminate, Gravol, TripTone, Wal-Dram.
dimenhydrinate is illustrative MVP content compiled from public sources. pharmacopeia is for educational and informational use only and is not a substitute for professional medical advice.